Khaled Essa
gast promovemdus
- Naam
- K.T.S.E.M. Essa
- Telefoon
- 071 5274324
- k.t.s.e.m.essa@lacdr.leidenuniv.nl
For more information look at the English website
gast promovemdus
- Faculteit der Wiskunde en Natuurwetenschappen
- LACDR
- Divisie Medicinal Chemistry
Promovendus
- Faculteit der Wiskunde en Natuurwetenschappen
- LACDR
- Divisie Medicinal Chemistry
- Essa K.T.S.E.M., Noorman Dussen K. van der, Yao Y., Bleijs B.T.M., Ortiz Zacarias N.V., Heitman L.H., Westen G.J.P. van, Jespers W., Es D. van der & Sicho M. (2025), Combining AlphaFold with focused virtual library design in the development of novel CCR2 and CCR5 antagonists, Journal of Chemical Information and Modeling 65(22): 12398-12409.
- Essa K., Ortiz Zacarías N.V., Roth S., Xin B.T., Winter S. de, Horst C. van der, Bleijs B., Heiden R.A. de, Voulgaraki R., Neubert E., Ovaa H., Danen E.H.J., Mulder M.P.C., Moreau K., Es D. van der & Heitman L.H. (2025), Leveraging targeted protein degradation for G protein-coupled receptors: the development of CCR2 molecular degraders, Journal of Medicinal Chemistry 68(24): 26525-26546.