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Research
Determining the kinetic profile of ENT1 inhibitors
Science
Leiden Academic Centre for Drug Research (LACDR)
Drug Discovery & Safety
Medicinal Chemistry
Allosteric Modulation
Science
Leiden Academic Centre for Drug Research (LACDR)
Drug Discovery & Safety
Medicinal Chemistry
Better ligands for G Protein-Coupled Receptors
Science
Leiden Academic Centre for Drug Research (LACDR)
Drug Discovery & Safety
Medicinal Chemistry
Cannabinoid receptor 2 as a ‘drugable’ target: kinetic profile of novel receptor ligands
Science
Leiden Academic Centre for Drug Research (LACDR)
Drug Discovery & Safety
Medicinal Chemistry
Cheminformatics: Analyzing small-molecule activity data
Science
Leiden Academic Centre for Drug Research (LACDR)
Drug Discovery & Safety
Medicinal Chemistry
Covalent inhibitors of G protein-coupled receptors: the case of adenosine receptors
Science
Leiden Academic Centre for Drug Research (LACDR)
Drug Discovery & Safety
Medicinal Chemistry
Intracellular allosteric modulators for human CC chemokine receptors
Science
Leiden Academic Centre for Drug Research (LACDR)
Drug Discovery & Safety
Medicinal Chemistry
Inverse Agonism and Constitutive Activity
Science
Leiden Academic Centre for Drug Research (LACDR)
Drug Discovery & Safety
Medicinal Chemistry
Kinetic profiling of positive allosteric modulators of the mGlu2 receptor
Science
Leiden Academic Centre for Drug Research (LACDR)
Drug Discovery & Safety
Medicinal Chemistry
Kinetics for drug discovery – The first step towards an improved drug discovery paradigm
Science
Leiden Academic Centre for Drug Research (LACDR)
Drug Discovery & Safety
Medicinal Chemistry
Kinetics for Drug Discovery: a Case for the Adenosine A3 receptor
Science
Leiden Academic Centre for Drug Research (LACDR)
Drug Discovery & Safety
Medicinal Chemistry
Novel receptor concepts
Science
Leiden Academic Centre for Drug Research (LACDR)
Drug Discovery & Safety
Medicinal Chemistry
Personalized Medicine
Science
Leiden Academic Centre for Drug Research (LACDR)
Drug Discovery & Safety
Medicinal Chemistry
Receptor Residence Time
Science
Leiden Academic Centre for Drug Research (LACDR)
Drug Discovery & Safety
Medicinal Chemistry
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