Research output
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Dissertation Clavis Aurea? Structure-enabled approaches of identifying and optimizing GPCR ligands
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Science
- Leiden Academic Centre for Drug Research (LACDR)
- Drug Discovery & Safety
- Medicinal Chemistry
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Science
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Dissertation Transforming data into knowledge for intelligent decision-making in early drug discovery
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Science
- Leiden Academic Centre for Drug Research (LACDR)
- Drug Discovery & Safety
- Medicinal Chemistry
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Science
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Dissertation Allosteric modulation by sodium ions and amilorides of G protein-coupled receptors
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Science
- Leiden Academic Centre for Drug Research (LACDR)
- Drug Discovery & Safety
- Medicinal Chemistry
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Science
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Publication The Role of Target Binding Kinetics in Drug Discovery
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Science
- Leiden Academic Centre for Drug Research (LACDR)
- Drug Discovery & Safety
- Medicinal Chemistry
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Science
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Publication A large-scale crop protection bioassay data set
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Science
- Leiden Academic Centre for Drug Research (LACDR)
- Drug Discovery & Safety
- Medicinal Chemistry
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Science
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Publication Affinity and kinetics study of anthranilic acids as HCA2 receptor agonists
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Science
- Leiden Academic Centre for Drug Research (LACDR)
- Drug Discovery & Safety
- Medicinal Chemistry
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Science
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Publication Structure-affinity relationships (SARs) and structure-kinetics relationships (SKRs) of Kv11.1 blockers
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Science
- Leiden Academic Centre for Drug Research (LACDR)
- Drug Discovery & Safety
- Medicinal Chemistry
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Science
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Publication Structure-kinetics relationships of Capadenoson derivatives as adenosine A1 receptor agonists
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Science
- Leiden Academic Centre for Drug Research (LACDR)
- Drug Discovery & Safety
- Medicinal Chemistry
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Science
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Publication Whole-cell biosensor for label-free detection of GPCR-mediated drug responses in personal cell lines
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Science
- Leiden Academic Centre for Drug Research (LACDR)
- Drug Discovery & Safety
- Medicinal Chemistry
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Science
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Publication Evaluation of (4-Arylpiperidin-1-yl)cyclopentanecarboxamides As High-Affinity and Long-Residence-Time Antagonists for the CCR2 Receptor
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Science
- Leiden Academic Centre for Drug Research (LACDR)
- Drug Discovery & Safety
- Medicinal Chemistry
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Science
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Publication Indanes-Properties, Preparation, and Presence in Ligands for G Protein Coupled Receptors
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Science
- Leiden Academic Centre for Drug Research (LACDR)
- Drug Discovery & Safety
- Medicinal Chemistry
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Science
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Publication Mycobacterial dihydrofolate reductase inhibitors identified using chemogenomic methods and in vitro validation
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Science
- Leiden Academic Centre for Drug Research (LACDR)
- Drug Discovery & Safety
- Medicinal Chemistry
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Science
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Publication Scanning mutagenesis in a yeast system delineates the role of the NPxxY(x)(5,6)F motif and helix 8 of the adenosine A(2B) receptor in G protein coupling
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Science
- Leiden Academic Centre for Drug Research (LACDR)
- Drug Discovery & Safety
- Medicinal Chemistry
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Science
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Publication Proteochemometric modelling coupled to in silico target prediction
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Science
- Leiden Academic Centre for Drug Research (LACDR)
- Drug Discovery & Safety
- Medicinal Chemistry
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Science
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Publication Synthesis and biological evaluation of spirocyclic antagonists of CCR2 (chemokine CC receptor subtype 2)
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Science
- Leiden Academic Centre for Drug Research (LACDR)
- Drug Discovery & Safety
- Medicinal Chemistry
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Science